GDC046 Size:100 mg solid CFTR Inhibitor II inhibits SLC26A9-mediated
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GDC046 Size:100 mg solid CFTR Inhibitor II inhibits SLC26A9-mediatedGDC046 (Compound 3) is a potent, selective, and orally bioavailable inhibitor of TYK2 with Ki of 4. 8 nM, 83. 8 nM, 27. 6 nM and 253 nM for TYK2, JAK1, JAK2, and JAK3, respectively. Product information CAS Number: 1258292 64 6 Molecular Weight: 350. 20 Formula: C16H13Cl2N3O2 Chemical Name: 2, 6 dichloro N (2 (cyclopropanecarboxamido)pyridin 4 yl)benzamide Smiles: O=C(NC1=CC(NC(=O)C2CC2)=NC=C1)C1C(Cl)=CC=CC=1Cl InChiKey: IAFNAEGXTKTGHN UHFFFAOYSA N
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